PDB Entry - 5EDR

(Status - Released)

Summary information:

Title: EGFR kinase (T790M/L858R) with inhibitor compound 27: ~{N}-(1~{H}-indazol-3-yl)-7,7-dimethyl-2-(2-methylpyrazol-3-yl)-5~{H}-furo[3,4-d]pyrimidin-4-amine

PDB DOI: https://doi.org/10.2210/pdb5edr/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2015.11.078

Entry authors: Eigenbrot, C., Yu, C.

Initial deposition on: 21 October 2015

Initial release on: 2 December 2015

Latest revision on: 6 March 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

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