PDB Entry - 5DLX

(Status - Released)

Summary information:

Title: FIRST DOMAIN OF HUMAN BROMODOMAIN BRD4 IN COMPLEX WITH INHIBITOR N-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-1-{3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}piperidine-4-carboxamide

PDB DOI: https://doi.org/10.2210/pdb5dlx/pdb

Primary publication DOI: https://doi.org/10.1021/acschembio.6b00286

Entry authors: Raux, B., Rebuffet, E., Betzi, S., Morelli, X.

Initial deposition on: 7 September 2015

Initial release on: 1 June 2016

Latest revision on: 10 January 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

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