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Structural and Biochemical Basis for Development of Influenza Virus Inhibitors Targeting the PA Endonuclease

Figure 6

Reported IC50 values of 4-substituted 2,4-dioxobutanoic acid inhibitors determined in an in vitro transcription assay with influenza A polymerase.

aPublished results in an influenza virus in vitro transcription assay [15]. bPublished results in an influenza virus in vitro transcription assay [26].

Figure 6

doi: https://doi.org/10.1371/journal.ppat.1002830.g006