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Synthesis of [1,3]Thiazolo[2,3-i]purinium Systems

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Abstract

The alkylation of purine-6-thiol with methallyl chloride and propargyl bromide in aqueous alcohol in the presence of alkali gave 6-[methallyl(propargyl)sulfanyl]purines which reacted with iodine and bromine to afford fused [1,3]thiazolo[2,3-i]purinium systems.

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Correspondence to K. Yu. Osheko.

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Original Russian Text © K.Yu. Osheko, D.G. Kim, O.S. El’tsov, T.S. Shtukina, 2018, published in Zhurnal Organicheskoi Khimii, 2018, Vol. 54, No. 9, pp. 1390–1394.

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Osheko, K.Y., Kim, D.G., El’tsov, O.S. et al. Synthesis of [1,3]Thiazolo[2,3-i]purinium Systems. Russ J Org Chem 54, 1406–1410 (2018). https://doi.org/10.1134/S1070428018090233

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  • DOI: https://doi.org/10.1134/S1070428018090233

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