Abstract
A diphenylmethyl protective group is suggested for use in the synthesis of 5-R-3-nitro-1H-1,2,4-triazoles unsubstituted at the cyclic nitrogen atom, via nucleophilic substitution of 5-bromo- and 5-methylsulfonyl groups.
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Tolstyakov, V.V., Tselinskii, I.V. Diphenylmethyl Protective Group in the Synthesis of 5-Substituted 3-Nitro-1H-1,2,4-triazoles. Russian Journal of General Chemistry 74, 399–404 (2004). https://doi.org/10.1023/B:RUGC.0000030397.19585.ec
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DOI: https://doi.org/10.1023/B:RUGC.0000030397.19585.ec