Research paperStructure–activity relationships for lipoprotein lipase agonists that lower plasma triglycerides in vivo
Under a Creative Commons license
open access
Graphical abstract
Keywords
Lipoprotein lipase
LPL
Triglyceride
Structure–activity relationship
Agonist
Abbreviations
ADME
absorption, distribution, metabolism and excretion
ANGPTL
angiopoietin-like protein
apo-
apolipoprotein
BINOL
1,1′-bi-2-naphthol
BSA
bovine serum albumin
CAD
coronary artery disease
EC50
effective concentration 50%
LPL
lipoprotein lipase
SAR
structure activity relationship
TG
triacylglycerol
VLDL
very low density lipoprotein
Cited by (0)
Copyright © 2015 The Authors. Published by Elsevier Masson SAS