General Pharmacology: The Vascular System
Volume 26, Issue 5, September 1995, Pages 911-944
ReviewThe mammalian tachykinin receptors
References (279)
- et al.
Antitussive effect of SR 48,968, a nonpeptide tachykinin NK2 receptor antagonist
Eur. J. Pharmac.
(1993) - et al.
Neurokinin A (NK2) receptor revisited with SR 48,968 a potent nonpeptide antagonist
Biochem. biophys. Res. Commun.
(1992) - et al.
Pharmacologic characterization of the novel ligand [4,5-3H-Leu]neurokinin A binding to NK2 receptors on hamster urinary bladder
Neuropeptides
(1992) - et al.
Calcium influx and protein kinas Ca activation mediate arachidonic acid mobilization by the human NK2 receptor expressed in CHO cells
FEBS Lett.
(1994) - et al.
The presence of NK-3 tachykinin receptors on rat uterus
Eur. J. Pharmac.
(1991) - et al.
Functional nonequivalence of structurally homologous domains of NK1 and NK2 type tachykinin receptors
J. biol. Chem.
(1993) - et al.
The rational development of small molecule tachykinin NK receptor selective antagonist-the utilisation of a dipeptide chemlical library in drug design
Bioorg. med. Chem. Lett.
(1994) - et al.
In vivo evidence for the activation of a septide-sensitive tachykinin receptor in guinea-pig bronchoconstriction
Life Sci. Pharmac. Lett.
(1994) - et al.
Antiemetic profile of a nonpeptide neurokinin NK1 receptor antagonist, CP 99,994 in ferrets
Eur. J. Pharmac.
(1993) - et al.
Rational design of high affinity tachykinin NK1 receptor antagonists
Bioorg. med. Chem.
(1994)
Rational design of high affinity tachykinin NK2 receptor antagonists
Bioorg. med. Chem.
(1994)
[125]His-NKA binds selectively to NK2 receptors of the B-type in rat small intestine smooth muscle membrane
Eur. J. Pharmac.
(1992)
Evidence for tachykinin NK2B-like receptors in guinea-pig alveolar macrophages
Life Sci. Pharmac. Lett.
(1992)
Molecular characterisation expression and localization of human NK3 receptor
FEBS Lett.
(1992)
Septide but not substance P stimulates inhibitory neurons in guinea-pig ileum
Eur. J. Pharmac.
(1994)
Characterization of the interaction of N-acyl-L-Trp benzyl ester neurokinin antagonists with the human NK1 receptor
J. biol. Chem.
(1994)
The effect of intrathecal administration of RP 67,580, a potent NK1 antagonist on nociceptive transmission in the rat spinal cord
Neurosci. Lett.
(1993)
Selective agonists of NK-2 binding sites highly active on rat portal vein (NK3 bioassay)
Neuropeptides
(1991)
[Pro9]SP and [pGlu6, Pro9]SP(6-11) interact with two different receptors in the guinea-pig ileum as demonstrated with new SP antagonists
Neuropeptides
(1992)
The nonpeptide tachykinin NK2 receptor antagonist SR 48,968 interacts with human but not rat cloned NK3 receptors
Biochem. biophys. Res. Commun.
(1994)
Characterization of neurokinin receptors in various isolated organs by the use of selective agonists
Life Sci.
(1987)
Specific agonists for neurokinin B receptors
Eur. J. Pharmac.
(1987)
Direct evidence that capsaicin-induced plasma protein extravasation is mediated through tachykinin NK1 receptors
Eur. J. Pharmac.
(1991)
Pharmacological examination of receptors mediating contractile responses to TKs in airways isolated from human, guineapig and hamster
J. Pharmac. exp. Ther.
(1993)
Active polypeptides of the amphibian skin and their synthetic analogs
Pure appl. Chem.
(1973)
Species differences between [3H] substance P binding in rat and guinea-pig shown by the use of peptide agonists and antagonists
Eur. J. Pharmac.
(1991)
Distribution and characterization of tachykinin binding in bronchopulmonary tract of rat and guinea-pig
Regul. Peptides
(1992)
In vitro pharmacological properties of RPR 100,893, a novel nonpeptide antagonist of the human NK1 receptor
Neuropeptides
(1994)
The involvement of neurokinin receptor subtypes in somatosensory processing in the superficial dorsal horn of the cat
Brain Res.
(1990)
Localization of agonist and antagonist binding domains of the human NK1 receptor
J. biol. Chem.
(1992)
Molecular bases for the species selectivity of the NK1 receptor antagonists CP 96,345 and RP 67,580
J. biol. Chem.
(1992)
The role of Histidine 265 in antagonist binding to the NK1 receptor
J. biol. Chem.
(1994)
A novel substance P binding site in bovine adrenal medulla
Neurosci. Lett.
(1990)
The human neurokinin A (substance K) receptor
J. biol. Chem.
(1990)
Molecular aspects of the tachykinin receptors
Regul. Peptides
(1993)
Chimeric NK1 (Substance P)/NK3 (neurokinin B) receptors
J. biol. Chem.
(1993)
Species differences in affinities of nonpeptide antagonists for substance P receptors
Eur. J. Pharmac.
(1991)
Activity at phencyclidine and mu opioid sites mediates the hyperalgesic and antinociceptive properties of the N-terminus of SP in a model of visceral pain
Neuroscience
(1994)
Molecular cloning of substance P cDNA from guinea-pig uterus
Biochim. biophys Acta
(1992)
Isolation and characterization of the human lung NK2 receptor gene using rapid amplification of cDNA ends
Biochem. biophys. Res. Commun.
(1991)
Tachykinin receptor types: classification and membrane signalling mechanisms
Neurochem. Int.
(1991)
[125I]NKA labels pharmacologically distinct populations of NK2 binding sites in hamster and rabbit urinary bladder
Eur. J. Pharmac.
(1993)
Vineyard peptide conference bears fruit
Trends Pharmac. Sci.
(1993)
Receptor-selective, peptidase-resistant agonists at NK1 and NK2 receptors: new tools for investigating neurokinin function
Neuropeptides
(1991)
Pharmacologic characterization of binding of the novel ligand [4,5-3HLeu9]NKA to NK2 receptors on hamster urinary bladder
FASEB J.
(1992)
Pharmacological characterization of cloned human NK2 (neurokinin A) receptor expressed in a baculovirus /Sf-21 insect cell system
Molec. Pharmac.
(1993)
Isolation and pharmacological characterization of a hamster urinary bladder neurokinin A receptor cDNA
Molec. Pharmac.
(1994)
Characterization of the tachykinin NK2 receptor in human bronchus: influence of amastatin-sensitive metabolic pathways
Br. J. Pharmac.
(1994)
In vitro and in vivo pharmacology of the non peptide antagonist at tachykinin NK2 receptors, GR 159,897
Br. J. Pharmac.
(1994)
Nonpeptide antagonists, CP 96,345 and RP 67,580, distinguish species variants in tachykinin NK2 receptors
Br. J. Pharmac.
(1993)
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