Skip to main content
SpringerLink
Log in

Search for novel, high affinity histamine H3 receptor ligands with fluorescent properties

  • Short Communication
  • Published:
Inflammation Research Aims and scope Submit manuscript

This is a preview of subscription content, log in via an institution to check access.

Access this article

Log in via an institution

Price excludes VAT (USA)
Tax calculation will be finalised during checkout.

Instant access to the full article PDF.

Institutional subscriptions

Fig. 1
Fig. 2

References

  1. Stark H, Kathmann M, Schlicker E, Schunack W, Schlegel B, Sippl W. Medicinal chemical and pharmacological aspects of imidazole-containing histamine H3 receptor antagonists. Mini Rev Med Chem. 2004;4:965–77.

    CAS  PubMed  Google Scholar 

  2. Cowart M, Altenbach R, Black L, Faghih R, Zhao C, Hancock AA. Medicinal chemistry and biological properties of non-imidazole histamine H3 antagonists. Mini Rev Med Chem. 2004;4:979–92.

    CAS  PubMed  Google Scholar 

  3. McGrath JC, Arribas S, Daly CJ. Fluorescent ligands for the study of receptors. Trends Pharmacol Sci. 1996;17:393–9.

    Article  CAS  PubMed  Google Scholar 

  4. Kuder K, Kieć-Kononowicz K. Fluorescent GPCR ligands as new tools in pharmacology. Curr Med Chem. 2008;21:2132–43.

    Article  Google Scholar 

  5. Amon M, Ligneau X, Camelin J-C, Berrebi-Bertrand I, Schwartz J-C, Stark H. Highly potent fluorescence-tagged non-imidazole histamine H3 receptor ligands. ChemMedChem. 2007;2:708–16.

    Article  CAS  PubMed  Google Scholar 

  6. Lesyk R, Zimenkovsky B, Subtelna I, Nektegayev I, Kazmirchuk G. Synthesis and antiinflammatory activity of some 2-arylamino-2-thiazoline-4-ones. Act Pol Pharm Drug Res. 2003;60:457–66.

    CAS  Google Scholar 

Download references

Acknowledgments

The work is partly supported by the Ministry of Scientific Research and Information Technology, Poland grant No. DAAD/55/2007, and the DAAD Germany (PPP Polen D/06/25529). Authors acknowledge ABL&E JASCO Poland for evaluation the fluorescent properties of 5. K. J. Kuder, T. Kottke, H. Stark, R. Seifert, and K. Kieć-Kononowicz are affiliated with COST Action BM0806.

Author information

Authors and Affiliations

  1. Department of Technology and Biotechnology of Drugs, Collegium Medicum, Jagiellonian University, Medyczna Str. 9, 30-688, Kraków, Poland

    K. J. Kuder & K. Kieć-Kononowicz

  2. Institut für Pharmazeutische Chemie, Johann Wolfgang Goethe Universität, Biozentrum, ZAFES/LiFF/CMP, Max-von-Laue-Str. 9, 60438, Frankfurt am Main, Germany

    T. Kottke & H. Stark

  3. Bioprojet Biotech, 4 rue Chesnay Beauregard, 35762, Saint Gregorie Cedex, France

    X. Ligneau & J.-C. Camelin

  4. Medical School of Hannover, Institute of Pharmacology, Carl-Neuberg-Str. 1, 30625, Hannover, Germany

    R. Seifert

Authors
  1. K. J. Kuder
    View author publications

    You can also search for this author in PubMed Google Scholar

  2. T. Kottke
    View author publications

    You can also search for this author in PubMed Google Scholar

  3. H. Stark
    View author publications

    You can also search for this author in PubMed Google Scholar

  4. X. Ligneau
    View author publications

    You can also search for this author in PubMed Google Scholar

  5. J.-C. Camelin
    View author publications

    You can also search for this author in PubMed Google Scholar

  6. R. Seifert
    View author publications

    You can also search for this author in PubMed Google Scholar

  7. K. Kieć-Kononowicz
    View author publications

    You can also search for this author in PubMed Google Scholar

Corresponding author

Correspondence to K. Kieć-Kononowicz.

Rights and permissions

Reprints and permissions

About this article

Cite this article

Kuder, K.J., Kottke, T., Stark, H. et al. Search for novel, high affinity histamine H3 receptor ligands with fluorescent properties. Inflamm. Res. 59 (Suppl 2), 247–248 (2010). https://doi.org/10.1007/s00011-009-0142-3

Download citation

  • Published:

  • Issue Date:

  • DOI: https://doi.org/10.1007/s00011-009-0142-3

Keywords

Search

Navigation