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A new intermediate for the rapid synthesis of N-isopropyl-p-/125I/- or p-/123I/ amphetamine

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Abstract

The triazene derivative of N-isopropylamphetamine XI, has been prepared in seven steps from amphetamine, as a new intermediate which is readily converted to N-isopropyl-p-iodoamphetamine /XII/. XI makes now possible the simple, rapid and regiospecific synthesis of /125I/- or /123I/-XII direct before the application.

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Authors and Affiliations

  1. Department of Organic Chemistry, Charles University, Albertov 2030, 128 40, Prague 2, Czechoslovakia

    J. Protiva, V. Křeček & L. Lešetický

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  1. J. Protiva
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  2. V. Křeček
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  3. L. Lešetický
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Protiva, J., Křeček, V. & Lešetický, L. A new intermediate for the rapid synthesis of N-isopropyl-p-/125I/- or p-/123I/ amphetamine. Journal of Radioanalytical and Nuclear Chemistry Letters 107, 331–336 (1986). https://doi.org/10.1007/BF02164198

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  • DOI: https://doi.org/10.1007/BF02164198

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