Skip to main content
SpringerLink
Log in

Reagents for new heteroannelation reactions III. 2-(Methylthio)-2-thiazoline

Reagentien für neue Heteroanellierungsreaktionen, 3. Mitt. 2-(Methylthio)-2-thiazolin

  • Organische Chemie Und Biochemie
  • Published:
Monatshefte für Chemie / Chemical Monthly Aims and scope Submit manuscript

Summary

A variety of partly novel tri- and tetracyclic hetero systems were obtained by reaction of heteroaromatic 2-aminoesters with 2-(methylthio)-2-thiazoline, yielding double-annelation of a thiazolo[2,3-b]pyrimido moiety in a one-pot process.

Zusammenfassung

Eine Reihe z.T. neuer tri- und tetracyclischer Heterosysteme wurde durch Reaktion von heteroaromatischen 2-Aminoestern mit 2-(Methylthio)-2-thiazolin erhalten, wobei im Eintopfverfahren durch doppelte Cyclisierung jeweils eine Thiazolo[2,3-b]pyrimido-Einheit anelliert wurde.

This is a preview of subscription content, log in via an institution to check access.

Access this article

Log in via an institution

Price excludes VAT (USA)
Tax calculation will be finalised during checkout.

Instant access to the full article PDF.

Institutional subscriptions

Similar content being viewed by others

References

  1. Part II: Sauter F, Fröhlich J, Chowdhury AZMS, Hametner C (1996) Acta Chim Slov (in press)

  2. Sauter F, Fröhlich J, Blasl K, Gewald K (1995) Heterocyles40: 851

    Google Scholar 

  3. Sauter F, Fröhlich J, Ahmed EK (1996) Monatsh Chem127: 319

    Google Scholar 

  4. Jansen JE (1942) US Patent 2, 293,465

  5. Bose AK, Fahey JL, Manhas MS (1973) J Heterocycl Chem10: 791

    Google Scholar 

  6. Sauter F, Deinhammer W (1974) Monatsh Chem105: 452

    Google Scholar 

  7. Sauter F, Deinhammer W, Danksagmüller K (1974) Monatsh Chem105: 863

    Google Scholar 

  8. Sauter F, Deinhammer W, Danksagmüller K (1974) Monatsh Chem105: 882

    Google Scholar 

  9. Sauter F, Deinhammer W, Stanetty P (1974) Monatsh Chem105: 1258

    Google Scholar 

  10. Chern JW, Liu KC, Shish FJ, Chan CH (1987) Arch Pharm320: 1276

    Google Scholar 

  11. Svetlik J (1987) Liebigs Ann Chem1987: 1121

    Google Scholar 

  12. Manhas MS, Amin SG (1976) J Heterocylc Chem13: 903

    Google Scholar 

  13. Howe RK, Bolluyt SC (1969) J Org Chem34: 1713

    Google Scholar 

  14. Schmidt P, Eichenberger K, Wilhelm M, Druey J (1959) Helv Chim Acta42: 349

    Google Scholar 

  15. Shvedov VI, Ryzhkova VK, Grinev AN (1967) Khim Geterosikl Soedin1967: 1010

    Google Scholar 

  16. Pregnolato M, Borgna P, Terreni M (1995) J Heterocycl Chem32: 847

    Google Scholar 

  17. Gompper R, Gaeng M, Saygin F (1966) Tetrahedron Lett1966: 1885

    Google Scholar 

  18. Gewald K, Blauschmidt P, Mayer R (1967) J Prakt Chem35: 97

    Google Scholar 

  19. Gewald K, Schinke E, Böttcher H (1966) Chem Ber99: 94

    Google Scholar 

  20. Ahmed EK (1995) Monatsh Chem126: 953

    Google Scholar 

  21. Kato Y (1972) Yakugaku Zasshi93: 397

    Google Scholar 

  22. Perrissin M, Luu Doc C, Narcisse G, Bakri-Logeais F, Huguet F (1980) Eur J Med Chem Chim Ther15: 413

    Google Scholar 

  23. Arya VP (1972) Ind J Chem10: 1141

    Google Scholar 

Download references

Author information

Authors and Affiliations

  1. Institute of Organic Chemistry, Vienna University of Technology, A-1060, Vienna, Austria

    F. Sauter, J. Fröhlich, A. Z. M. S. Chowdhury & C. Hametner

Authors
  1. F. Sauter
    View author publications

    You can also search for this author in PubMed Google Scholar

  2. J. Fröhlich
    View author publications

    You can also search for this author in PubMed Google Scholar

  3. A. Z. M. S. Chowdhury
    View author publications

    You can also search for this author in PubMed Google Scholar

  4. C. Hametner
    View author publications

    You can also search for this author in PubMed Google Scholar

Additional information

Dedicated to pharmacistT. Mayrhofer, the long-standing sponsor of pharmaceutical research, on the occasion of his 90th birthday

On leave from University of Chittagong, Bangladesh

Rights and permissions

Reprints and permissions

About this article

Cite this article

Sauter, F., Fröhlich, J., Chowdhury, A.Z.M.S. et al. Reagents for new heteroannelation reactions III. 2-(Methylthio)-2-thiazoline. Monatsh Chem 128, 503–508 (1997). https://doi.org/10.1007/BF00806858

Download citation

  • Received:

  • Accepted:

  • Issue Date:

  • DOI: https://doi.org/10.1007/BF00806858

Keywords

Search

Navigation