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Purines and pyrimidines and condensed systems based on them. 2. Synthesis of 1-methyl-9-aminoxanthine and 9-aminotheophylline

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

The previously unknown 9-aminotheophylline and 1-methyl-9-aminoxanthine were synthesized from 3-methyl-5-amino-6-hydrazinouracil. In the case of 1-methyl-9-aminoxanthine an x-ray diffraction study of an N-amino derivative of an NH heterocycle was made for the first time.

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Authors and Affiliations

  1. Scientific-Research Institute of Physical and Organic Chemistry, Rostov State University, Rostov-on-Don

    V. V. Kuz'menko, T. A. Kuz'menko, G. G. Aleksandrov, A. F. Pozharskii & A. V. Gulevskaya

  2. M. A. Suslov Rostov State University, 344006, Rostov-on-Don

    V. V. Kuz'menko, T. A. Kuz'menko, G. G. Aleksandrov, A. F. Pozharskii & A. V. Gulevskaya

Authors
  1. V. V. Kuz'menko
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  2. T. A. Kuz'menko
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  3. G. G. Aleksandrov
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  4. A. F. Pozharskii
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  5. A. V. Gulevskaya
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Additional information

See [1] for communication 1.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 6, pp. 836–844, June, 1987.

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Kuz'menko, V.V., Kuz'menko, T.A., Aleksandrov, G.G. et al. Purines and pyrimidines and condensed systems based on them. 2. Synthesis of 1-methyl-9-aminoxanthine and 9-aminotheophylline. Chem Heterocycl Compd 23, 690–697 (1987). https://doi.org/10.1007/BF00486922

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  • DOI: https://doi.org/10.1007/BF00486922

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