Abstract
Cyclization of arylhydrazones to indoles.
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References
(a) Fischer, E.; Jourdan, F. Ber. 1883, 16, 2241–2245. H. Emil Fischer (1852–1919) is arguably the greatest organic chemist ever. He was born in Euskirchen, near Bonn, Germany. When he was a boy, his father, Lorenz, said about him: “The boy is too stupid to go in to business; so in God’s name, let him study.” Fischer studied at Bonn and then Strassburg under Adolf von Baeyer. Fischer won the Nobel Prize in Chemistry in 1902 (three years ahead of his master, von Baeyer) for his synthetic studies in the area of sugar and purine groups. Sadly, Fischer committed suicide after WWI after his son died during the war and his fortunes completely gone. (b) Fischer, E.; Hess, O. Ber. 1884, 17, 559.
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Li, J.J. (2014). Fischer indole synthesis. In: Name Reactions. Springer, Cham. https://doi.org/10.1007/978-3-319-03979-4_106
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