Coating Processes of Pharmaceutical Applicability: A Glimpse
GLIMPSE ON PHARMACEUTICAL COATING PROCESSES
Abstract
Presentation of manuscript is aiming to furnish glimpse on coating processes. Coating is process of snugly covering substrate surface with coating materials (CoM). In due course coating process has gradually developed from sugar-coating to non-aqueous film-coating to aqueous film-coating to specialised-coating processes. In second half of past century sugar-coating was first choice for pharmaceutical industry. Lengthy and tedious processing along with issues of skilled-operator inherited to sugar-coating compelled them to spring-up and improve film-coating. From past five decades, volatile organic solvent (VOS) are preferred over water in film-coating. Momentum for using aqueous solvent in film-coating gets accelerated from past few decades. Nowadays these replacing the VOS based film-coating processes as later inherit issues relating toxicity; safety; worker hygiene & safety; environmental pollution; etc. During process of finding novelty of coating another exploited sphere is coating of particulate substrate surfaces with CoM is to confer them worthy functionalities and applications. In this area both wet- & dry-coating process finds applicability thru modifying and/or altering innate properties of substrate, physically and/or chemically. Dry-coating process basically comprises specialised and novel process & technologies. Nowadays there available numerous conventional, specialised, and novel coating processes. Amongst them state-of-art process are hot-melt coating (HMC) process, aqueous film-coating process, aerosolized coating process, Supercell® coating process, gas-/ vapour-phase process, photo curable coating process, electrical-electrostatic deposition process, Resonant acoustic coating process, thermal and mechanical process, thermo-mechanical process, fluidised-bed processes, etc. Herein conventional, specialised, and novel coating processes are briefed, to update professionals.
Keywords: Coating, film-coating, novel, process, specialised.
Keywords:
Coating, film-coating, novel, process, specialised
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References
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4. Nakamura S, Sakamoto T, Ito T, Kabasawa K, Yuasa H. Preparation of controlled-release fine particles using a dry coating method. AAPS PharmSciTech, 2016; 17:1393–1403.
5. Saikh MAA, Aqueous film coating the current trend. Journal of Drug Delivery and Therapeutics, 2021; 11(4-s):212-224. DOI: https://dx.doi.org/10.22270/jddt.v11i4-S.4911.
6. Ahmed SAN, Patil SR, Khan MKS, Khan MS. Tablet coating techniques: Concept and recent trends. International Journal of Pharmaceutical Sciences Review and Research, 2021; 66(1):43-53.
7. Arora R, Rathore KS, Bharkatiya M. An overview on tablet coating. Asian Journal of Pharmaceutical Research and Development, 2019; 7(4):89-92. DOI: http://dx.doi.org/10.22270/ajprd.v7i4.547.
8. Zaid AN. A Comprehensive review on pharmaceutical film coating: Past, present, and future. Drug Design Development and Therapy, 2020; 14:4613-4623.
9. Seo KS, Bajracharya R, Lee SH, Han HK. Pharmaceutical application of tablet film coating. Pharmaceutics, 2020; 12(9):853. DOI: http://dx.doi.org/10.3390/pharmaceutics12090853.
10. Saikh MAA. Film former in film coating. International Journal of Pharmaceutical Sciences and Research, 2022; 13(4): [In press]
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12. Saikh MAA, Mohapatra P. Thermo-mechanical dry coating as dry coating process is for pharmaceutical. Journal of Drug Delivery and Therapeutics, 2021; 11(6):176-187. DOI: https://dx.doi.org/10.22270/jddt.v11i6.5107.
13. Singhai NJ, Rawal A, Maurya R, Suman R. Design and characterization of dual drug loaded microspheres for colon drug targeting. Journal of Drug Delivery and Therapeutics, 2019; 9(3-s):12-22. DOI: https://dx.doi.org/10.22270/jddt.v9i3-s.2923.
14. Gaware RU, Tambe ST, Dhobale SM, Jadhav SL. Formulation and in-vitro evaluation of theophylline sustained release tablet. Journal of Drug Delivery and Therapeutics, 2019; 9(1-s):48-51. DOI: https://dx.doi.org/10.22270/jddt.v9i1-s.2252.
15. Saikh MAA. Dry coating of pharmaceutical powders. International Journal of Pharmaceutical Sciences and Research, 2022; 13(7): [In press]
16. Saikh MAA, Mohapatra P. Specialised coating processes finding pharmaceutical applicability. Journal of Drug Delivery and Therapeutics, 2021; 11(6):209-224. DOI: https://dx.doi.org/10.22270/jddt.v11i6.5133.
17. Pundir K, Parashar B. The innovations in tablet coating: A review. International Educational Applied Research Journal, 2019; 3(6):18-23.
18. Yang Q, Yuan F, Xu L, Yan Q, Yang Y, Wu D, Guo F, Yang G. An update of moisture barrier coating for drug delivery. Pharmaceutics, 2019; 11(9):436. DOI: https://dx.doi.org/10.3390/pharmaceutics11090436.
19. Yang Q, Ma Y, Zhu J. Dry powder coated osmotic drug delivery system. European Journal of Pharmaceutical Sciences, 2018; 111:383-392. DOI: https://dx.doi.org/10.1016/j.ejps.2017.10.001.
20. Foppoli AA, Maroni A, Cerea M, Zema L, Gazzaniga A. Dry coating of solid dosage forms: An overview of processes and applications. Drug Development and Industrial Pharmacy, 2017; 43(12):1919-1931.
21. Bungert N, Kobler M, Scherließ R. In-depth comparison of dry particle coating processes used in dpi particle engineering. Pharmaceutics, 2021; 13(4):580. DOI: https://dx.doi.org/10.3390/pharmaceutics13040580.
22. Sharma R, Setia G. Mechanical dry particle coating on cohesive pharmaceutical powders for improving flowability - A review. Powder Technology, 2019; 356:458-479, DOI: https://dx.doi.org/10.1016/j.powtec.2019.08.009.
23. Zhang R, Hoffmann T, Tsotsas E. Novel technique for coating of fine particles using fluidized bed and aerosol atomizer. Processes, 2020; 8:1525. DOI: https://dx.doi.org/10.3390/pr8121525.
24. Bannow J, Koren L, Salar-Behzadi S, Löbmann K, Zimmer A, Rades T. Hot melt coating of amorphous Carvedilol. Pharmaceutics, 2020; 12(6):519. DOI: https://dx.doi.org/10.3390/pharmaceutics12060519.
25. Salar-Behzadi S, Corzo C, Gomes Lopes D, Meindl C, Lochmann D, Reyer S. Novel approach for overcoming the stability challenges of lipid-based excipients. Part 2: Application of polyglycerol esters of fatty acids as hot melt coating excipients. European Journal of Pharmaceutics and Biopharmaceutics, 2020; 148:107-117. DOI: https://dx.doi.org/10.1016/j.ejpb.2020.01.009.
26. Salar-Behzadi S, Corzo C, Schaden L, Laggner P, Zimmer A. Correlation between the solid state of lipid coating and release profile of API from hot melt coated microcapsules. International Journal of Pharmaceutics, 2019; 565:569-578. DOI: https://dx.doi.org/10.1016/j.ijpharm.2019.05.036.
27. Stocker E, Becker K, Hate S, Hohl R, Schiemenz W, Sacher S, Zimmer A, Salar-Behzadi S. Application of ICH Q9 quality risk management tools for advanced development of hot melt coated multiparticulate systems. Journal of Pharmaceutical Sciences, 2017; 106(1):278-290. DOI: https://dx.doi.org/10.1016/j.xphs.2016.09.025.
28. Zier KI, Schultze W, Leopold CS. Combination of a hot-melt subcoating and an enteric coating for moisture protection of hygroscopic Sennae fructus tablets. Pharmaceutical Development and Technology, 2019; 24(10):1210-1217. DOI: https://dx.doi.org/10.1080/10837450.2019.1648509.
29. Wang X, Wang P, Huang C, Lin X, Gong H, He H, Cai C. Hot-melt sub- and outer coating combined with enteric aqueous coating to improve the stability of aspirin tablets. Asian Journal of Pharmaceutical Sciences, 2017; 12(3):266-278. DOI: https://dx.doi.org/10.1016/j.ajps.2016.11.003.
30. Guimarães TF, Comelli ACC, Tacón LA, Cunha TA, Marreto RN, Freitas LAP. Fluidized bed hot melt granulation with hydrophilic materials improves Enalapril maleate stability. AAPS PharmSciTech, 2017; 18(4):1302-1310. DOI: https://dx.doi.org/10.1208/s12249-016-0593-0.
31. Schertel S, Salar-Behzadi S, Karrer J, Laggner P, Zimmer A. Impact of polysorbate 65 on tripalmitin crystal growth and release stability of hot melt coated multiparticulate systems. International Journal of Pharmaceutics, 2021; 607:120970. DOI: https://dx.doi.org/10.1016/j.ijpharm.2021.120970.
32. Schertel S, Salar-Behzadi S, Zimmer A. Impact of surface properties of core material on the stability of hot melt-coated multiparticulate systems. Pharmaceutics, 2021; 13(3):366. DOI: https://dx.doi.org/10.3390/pharmaceutics13030366.
33. Lopes DG, Salar-Behzadi S, Zimmer A. Designing optimal formulations for hot-melt coating. International Journal of Pharmaceutics, 2017; 533(2):357-363. DOI: https://dx.doi.org/10.1016/j.ijpharm.2017.08.086.
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Saikh MAA. Coating Processes of Pharmaceutical Applicability: A Glimpse. JDDT [Internet]. 15Mar.2022 [cited 27Apr.2024];12(2):126-38. Available from: https://jddtonline.info/index.php/jddt/article/view/5362
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