PDB Entry - 6PS9

(Status - Released)

Summary information:

Title: Crystal structure of BRD4 bromodomain 1 with N-methylpyrrolidin-2-one (NMP) derivative 17 (5-{2-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]ethyl}-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indol-1-one)

PDB DOI: https://doi.org/10.2210/pdb6ps9/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmc.2019.115157

Entry authors: Ilyichova, O.V., Scanlon, M.J.

Initial deposition on: 12 July 2019

Initial release on: 27 November 2019

Latest revision on: 11 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (PDF)

Validation report (XML)

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