PDB Entry - 5KTX

(Status - Released)

Summary information:

Title: CREBBP bromodomain in complex with Cpd59 ((S)-1-(3-((2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)amino)-1-(tetrahydrofuran-3-yl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)ethanone)

PDB DOI: https://doi.org/10.2210/pdb5ktx/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.6b01022

Entry authors: Murray, J.M., Noland, C.

Initial deposition on: 12 July 2016

Initial release on: 2 November 2016

Latest revision on: 6 March 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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