PDB Entry - 4MEP

(Status - Released)

Summary information:

Title: Crystal Structure of the first bromodomain of human BRD4 in complex with a 3-chloro-pyridone ligand

PDB DOI: https://doi.org/10.2210/pdb4mep/pdb

Primary publication DOI: https://doi.org/10.1021/jm4011302

Entry authors: Filippakopoulos, P., Picaud, S., Felletar, I., Martin, S., Fedorov, O., Vidler, L.R., Brown, N., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Weigelt, J., Bountra, C., Hoelder, S., Knapp, S., Structural Genomics Consortium (SGC)

Initial deposition on: 27 August 2013

Initial release on: 25 September 2013

Latest revision on: 20 September 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (mmCIF)

Validation report (XML)

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