PDB Entry - 4L53

(Status - Released)

Summary information:

Title: Crystal Structure of (1R,4R)-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1H-pyrazol-1-yl}cyclohexan-1-ol bound to TAK1-TAB1

PDB DOI: https://doi.org/10.2210/pdb4l53/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2013.06.054

Entry authors: Wang, J., Hornberger, K.R., Crew, A.P., Jestel, A., Maskos, K., Moertl, M.

Initial deposition on: 10 June 2013

Initial release on: 3 July 2013

Latest revision on: 28 February 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (mmCIF)

Validation report (XML)

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