PDB Entry - 4ER7

(Status - Released)

Summary information:

Title: Crystal Structure of human DOT1L in complex with inhibitor SGC0947

PDB DOI: https://doi.org/10.2210/pdb4er7/pdb

Primary publication DOI: https://doi.org/10.1038/ncomms2304

Entry authors: Wernimont, A.K., Tempel, W., Yu, W., Scopton, A., Li, Y., Nguyen, K.T., Vedadi, M., Bradner, J.E., Schapira, M., Arrowsmith, C.H., Edwards, A.M., Bountra, C., Brown, P.J., Structural Genomics Consortium (SGC)

Initial deposition on: 19 April 2012

Initial release on: 16 May 2012

Latest revision on: 28 February 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (XML)

Validation report (PDF)

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