ReviewBile acid transporters and regulatory nuclear receptors in the liver and beyond
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Keywords
Bile acids
Cholestasis
Fatty liver disease
Gallstones
Liver regeneration
Liver cancer
Abbreviations
6-ECDCA
6-ethylchenodeoxycholic acid
AE2
anion exchanger 2
ABCG5/8
cholesterol efflux pump, ATP-binding cassette, subfamily G, member 5/8
BA
bile acid
AMPK
AMP activated protein kinase
BCRP (ABCG2)
breast cancer resistance protein, ATP-binding cassette, subfamily G, member 2
BRIC
benign recurrent intrahepatic cholestasis
BSEP (ABCB11)
bile salt export pump
CAR (NR1I3)
constitutive androstane receptor
EGFR
epidermal growth factor receptor
FGF15/19
fibroblast growth factor 15/19
FXR (NR1H4)
farnesoid X receptor/bile acid receptor
GLP-1
glucagon like peptide 1
GR (NR3C1)
glucocorticoid receptor
HCC
hepatocellular carcinoma
HNF1α
hepatocyte nuclear factor 1 alpha
HNF4α (NR2A1)
hepatocyte nuclear factor 4 alpha
IBABP (FABP6, ILBP)
intestinal bile acid-binding protein, fatty acid-binding protein 6
ICP
intrahepatic cholestasis of pregnancy
IL6
interleukin 6
LCA
lithocholic acid
LRH-1 (NR5A2)
liver receptor homolog-1
LXRα (NR1H3)
liver X receptor alpha
MDR1 (ABCB1)
p-glycoprotein, ATP-binding cassette, subfamily B, member 1
Mdr2/MDR3 (ABCB4)
multidrug resistance protein 2 (rodents)/3 (human)
MRP2 (ABCC2)
multidrug resistance-associated protein 2, ATP-binding cassette, subfamily C, member 2
MRP3 (ABCC3)
multidrug resistance-associated protein 3, ATP-binding cassette, subfamily C, member 3
MRP4 (ABCC4)
multidrug resistance-associated protein 4, ATP-binding cassette, subfamily C, member 4
NAFLD
non-alcoholic fatty liver disease
NASH
non-alcoholic steatohepatitis
norUDCA
norursodeoxycholic acid
NR
nuclear receptor
NTCP (SLC10A1)
sodium/taurocholate cotransporting polypeptide, solute carrier family 10, member 1
OATP1A2 (SLCO1A2, OATP1, OATP-A, SLC21A3)
solute carrier organic anion transporter family, member 1A2
OATP1B1 (SLCO1B1, OATP2, OATP-C, SLC21A6)
solute carrier organic anion transporter family, member 1B1
OATP1B3 (SLCO1B3, OATP8, SLC21A8)
solute carrier organic anion transporter family, member 1B3
OSTαβ
organic solute transporter alpha/beta
PBC
primary biliary cirrhosis
PFIC
progressive familial intrahepatic cholestasis
PH
partial hepatectomy
PPARα (NR1C1)
peroxisome proliferator-activated receptor alpha
PPARγ (NR1C3)
peroxisome proliferator-activated receptor gamma
PSC
primary sclerosing cholangitis
PXR (NR1I2)
pregnane X receptor
RARα (NR1B1)
retinoic acid receptor alpha
RXRα (NR2B1)
retinoid X receptor alpha
SHP (NR0B2)
short heterodimer partner
SRC2
p160 steroid receptor coactivator
TGR5
G protein-coupled bile acid receptor
TNFα
tumor necrosis factor α
TPN
total parenteral nutrition
UDCA
ursodeoxycholic acid
VDR (NR1I1)
vitamin D receptor. Please note that for the convenience of better readability and clarity, abbreviations for transporters and nuclear receptors were capitalized throughout this article when symbols were identical for human and rodents
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Copyright © 2012 European Association for the Study of the Liver. Published by Elsevier B.V.